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CYM5442
Contact us for more batch information
CYM5442
Catalog No. T2026Cas No. 1094042-01-9
CYM5442 is an S1P agonist, targeting to Sphingosine.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $39 | In Stock | |
| 2 mg | $55 | In Stock | |
| 5 mg | $89 | In Stock | |
| 10 mg | $139 | In Stock | |
| 25 mg | $263 | In Stock | |
| 50 mg | $428 | In Stock | |
| 100 mg | $653 | In Stock | |
| 500 mg | $1,350 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | CYM5442 is an S1P agonist, targeting to Sphingosine. |
| Kinase Assay | HDAC activity is detected as described in the Colorimetric HDAC Activity Assay kit. Each reaction (100 μL) contains nuclear protein (50 μg) extract from leukaemia cells and HDAC substrate. To test the effect of HDACis, Chidamide (CS055) and MS-275 are added to the mixtures and incubated at 37°C for 1 h. The HDAC activities are measured by a microplate readers at 405 nm. The positive control (only nuclear extract and vehicle) is set as 100% and double-distilled water containing 10 μM Trichostatin A, a known strong HDACi, is used as a negative control and set as 0%[2]. |
| Molecular Weight | 409.48 |
| Formula | C23H27N3O4 |
| Cas No. | 1094042-01-9 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
| Solubility Information | DMSO: Slightly soluble  |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。 Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Dose Conversion
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