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Edg-2 receptor inhibitor 1
🥰Excellent
Catalog No. T4521Cas No. 1195941-38-8
Alias SAR-100842
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
Edg-2 receptor inhibitor 1
🥰Excellent
Purity: 99.69%
Catalog No. T4521Alias SAR-100842Cas No. 1195941-38-8
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $98 | In Stock | |
| 2 mg | $178 | In Stock | |
| 5 mg | $288 | In Stock | |
| 10 mg | $449 | In Stock | |
| 25 mg | $698 | In Stock | |
| 50 mg | $996 | In Stock | |
| 100 mg | $1,330 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $303 | In Stock |
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Purity:99.69%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM). |
| Targets&IC50 | Edg2 receptor:<0.1 μM |
| In vitro | Edg-2 receptor inhibitor 1 is an inhibitor of the endothelial differentiation gene receptor 2 (Edg-2, EDG2), which is activated by lysophosphatidic acid (LPA) and is also termed as LPA1 receptor, and is useful for the treatment of diseases such as atherosclerosis, myocardial infarction and heart failure, for example[1]. |
| Alias | SAR-100842 |
| Molecular Weight | 445.51 |
| Formula | C27H27NO5 |
| Cas No. | 1195941-38-8 |
| Smiles | N(C(=O)C1=CC(OCCC2=CC(C)=CC=C2)=C(OC)C=C1)C3(C(O)=O)CC=4C(C3)=CC=CC4 |
| Relative Density. | 1.28 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 83.3 mg/mL (186.98 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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