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G-Protein antagonist peptide acetate

Catalog No. TP1902L1 CAS TP1902L1

G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide acetate inhibits the activation of Gi or Go by M2 muscarinic cholinergic receptor (M2 mAChR) or of Gs by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis

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G-Protein antagonist peptide acetate Chemical Structure

G-Protein antagonist peptide acetate, CAS TP1902L1

Pack Size	Availability	Price/USD
1 mg	In stock	$ 139.00
2 mg	In stock	$ 233.00
5 mg	In stock	$ 365.00
10 mg	In stock	$ 581.00
25 mg	In stock	$ 919.00
50 mg	In stock	$ 1,250.00
100 mg	In stock	$ 1,690.00

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Purity: 98.06%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Molecular Weight	1153.33
Formula	C59H68N12O11S
CAS No.	TP1902L1

Storage

store at low temperature,keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Mukai H, et al. G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J Biol Chem. 1992;267(23):16237-16243.

Related compound libraries

This product is contained In the following compound libraries：

Peptide Compound Library Inhibitor Library Neurotransmitter Receptor Compound Library

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Keywords

G-Protein antagonist peptide acetate TP1902L1 GPCR/G Protein Neuroscience Adrenergic Receptor G Protein antagonist peptide acetate G-Protein antagonist peptide Acetate GProtein antagonist peptide acetate inhibitor inhibit

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