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GLPG2938

🥰Excellent
Catalog No. T9199Cas No. 2130996-00-6
Alias 1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea

GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and selective antagonist of S1P2.

GLPG2938

GLPG2938

🥰Excellent
Purity: 98.25%
Catalog No. T9199Alias 1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)ureaCas No. 2130996-00-6
GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and selective antagonist of S1P2.
Pack SizePriceAvailabilityQuantity
1 mg$76In Stock
5 mg$163In Stock
10 mg$289In Stock
25 mg$578In Stock
50 mg$833In Stock
100 mg$1,150In Stock
1 mL x 10 mM (in DMSO)$179In Stock
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Purity:98.25%
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Product Introduction

Bioactivity
Description
GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and selective antagonist of S1P2.
In vitro
GLPG2938 significantly prevents the S1P-mediated contraction at all tested concentrations[1].
In vivo
In all species ,GLPG2938 shows good pharmacokinetics, with long half-life,low clearance,and good bioavailability.
Alias1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea
Chemical Properties
Molecular Weight503.4
FormulaC20H19F6N7O2
Cas No.2130996-00-6
SmilesCCOc1cc(NC(=O)NCc2cc(C)c(nn2)-c2cn(C)nc2C(F)(F)F)cc(n1)C(F)(F)F
Relative Density.1.49 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 60 mg/ml (119.19 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM1.9865 mL9.9325 mL19.8649 mL99.3246 mL
5 mM0.3973 mL1.9865 mL3.9730 mL19.8649 mL
10 mM0.1986 mL0.9932 mL1.9865 mL9.9325 mL
20 mM0.0993 mL0.4966 mL0.9932 mL4.9662 mL
50 mM0.0397 mL0.1986 mL0.3973 mL1.9865 mL
100 mM0.0199 mL0.0993 mL0.1986 mL0.9932 mL

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