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GX 201
Catalog No. T9647Cas No. 1788071-27-1
GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $131 | In Stock | |
| 5 mg | $328 | In Stock | |
| 10 mg | $493 | In Stock | |
| 25 mg | $788 | In Stock | |
| 50 mg | $1,120 | In Stock | |
| 100 mg | $1,490 | In Stock | |
| 500 mg | $2,960 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $363 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7. |
| In vivo | GX 201 has a relatively long half-life in mice. GX 201 produces analgesia at a free plasma concentration about 3 times the IC50 for high-affinity channel block. GX 201 inhibits nociceptive responses induced by formalin and inflammatory pain caused by complete Freund’s adjuvant (CFA)[1]. |
| Alias | GX-201 |
| Molecular Weight | 563 |
| Formula | C25H27ClF4N2O4S |
| Cas No. | 1788071-27-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||
| Solubility Information | DMSO: 5.63 mg/mL (10 mM)  | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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