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pimpinellin
🥰Excellent
Catalog No. T5776Cas No. 131-12-4
Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity.
pimpinellin
🥰Excellent
Purity: 99.85%
Catalog No. T5776Cas No. 131-12-4
Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 28 € | In Stock | |
| 5 mg | 64 € | In Stock | |
| 10 mg | 107 € | In Stock | |
| 25 mg | 216 € | In Stock | |
| 50 mg | 353 € | In Stock | |
| 100 mg | 520 € | In Stock | |
| 200 mg | 740 € | In Stock |
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CitedSelect Batch
Purity:99.85%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity. |
| In vitro | Pimpinellin had potent cytotoxic activities against the three cell lines, with the IC50 values of 14.4?±?0.3?μM, 20.4?±?0.5?μM, and 29.2?±?0.6?μM, respectively. The mechanism of the antitumor action indicated that pimpinellin inhibited the growth of MGC-803 cells via the induction of tumor cell apoptosis, with apoptosis ratio of 27.44% after 72?h of treatment at 20?μM. |
| Molecular Weight | 246.22 |
| Formula | C13H10O5 |
| Cas No. | 131-12-4 |
| Smiles | COc1c(OC)c2ccc(=O)oc2c2ccoc12 |
| Relative Density. | 1.352 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 49 mg/mL (199.0 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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