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Tienilic Acid
🥰Excellent
Catalog No. T36125Cas No. 40180-04-9
Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
Tienilic Acid
🥰Excellent
Purity: 99.61%
Catalog No. T36125Cas No. 40180-04-9
Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $39 | In Stock | |
| 10 mg | $72 | In Stock | |
| 25 mg | $147 | In Stock | |
| 50 mg | $218 | In Stock | |
| 100 mg | $323 | In Stock | |
| 200 mg | $483 | In Stock | |
| 500 mg | $776 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $50 | In Stock |
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Purity:99.61%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity |
| In vivo | In female and male Sprague-Dawley rats, Tienilic Acid decreased blood pressure and serum uric acid at 30 mg/kg. Tienilic acid decreased slightly hemoglobin and increased S-GPT at 120 and 480 mg/kg. Tienilic Acid significantly increase the liver weight and serum magnesium concentration in male rats, while the liver weight of female rats increased only slightly. Tienilic Acid also induced unicellular necrosis of small groups of liver cells[2]. |
| Molecular Weight | 331.17 |
| Formula | C13H8Cl2O4S |
| Cas No. | 40180-04-9 |
| Smiles | C(=O)(C1=C(Cl)C(Cl)=C(OCC(O)=O)C=C1)C2=CC=CS2 |
| Relative Density. | 1.532g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | Acetone-d6: 250 mg/mL (754.90 mM), Sonication and heating to 80℃ are recommended. DMSO: ≥ 33.1 mg/mL | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
Acetone-d6
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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