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WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $52 | In Stock | |
2 mg | $75 | In Stock | |
5 mg | $117 | In Stock | |
10 mg | $178 | In Stock | |
25 mg | $352 | In Stock | |
50 mg | $523 | In Stock | |
100 mg | $757 | In Stock | |
1 mL x 10 mM (in DMSO) | $138 | In Stock |
Description | WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases. |
Targets&IC50 | MOZ:55 nM |
In vitro | MOZ-IN-3is an inhibitor of MOZ(IC50=55 nM). MOZ-IN-3 causes cell senescence(IC50=1.6 μM) and suppresses the proliferation(IC50=551 nM). |
Kinase Assay | Reactions are set up with Acetyl coenzyme A (AcCoA)(0.4 μM), N-terminal histone H4 peptide (sequence SGRGKGGKGLGKGGAKRHRKV-GGK-biotin)(50 nM), MOZ enzyme(10 nM), and an acetyl-lysine specific antibody (final dilution 1: 10000). |
Alias | MOZ-IN-3 |
Molecular Weight | 384.42 |
Formula | C20H17FN2O3S |
Cas No. | 2055397-18-5 |
Smiles | Cc1cc(cc(C(=O)NNS(=O)(=O)c2ccccc2)c1F)-c1ccccc1 |
Relative Density. | 1.307 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 45 mg/mL (117.06 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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