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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $253 | In Stock | |
5 mg | $520 | In Stock | |
10 mg | $743 | In Stock | |
25 mg | $1,150 | In Stock | |
50 mg | $1,550 | In Stock | |
100 mg | $1,980 | In Stock | |
1 mL x 10 mM (in DMSO) | $652 | In Stock |
Description | CMP8 is a selective ligand for estrogen receptor. CMP8 binds to the mutant estrogen receptor ligand binding domain (ERLBD). CMP8 has IC50 values of 29 nM , 41 nM, 1100 nM and 2200 nM for MGERα, MGRERα, hERα and hERβ, respectively. |
In vivo | CMP8 is dosed in male Balb-c mice (4 mg/kg, ip). In mammalian cells, the plasma concentration after 4 h is 1.5-fold its EC50. It has a Cmax of 0.5 μM after 30 min.[1][2] |
Molecular Weight | 528.08 |
Formula | C33H34ClNO3 |
Cas No. | 851107-28-3 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||||||||||||
Solubility Information | DMSO: 50 mg/mL (94.68 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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