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Iferanserin
Catalog No. T15552Cas No. 58754-46-4
Alias S-MPEC
Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease.
Iferanserin
Catalog No. T15552Alias S-MPECCas No. 58754-46-4
Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 25 mg | $1,400 | 6-8 weeks | |
| 50 mg | $1,820 | 6-8 weeks | |
| 100 mg | $2,500 | 6-8 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Iferanserin (S-MPEC) is a selective antagonist of the serotonin (5-HT) receptor with a specific affinity for 5-HT2A receptors, showing potential for the treatment of internal hemorrhoid disease. |
| In vitro | Iferanserin might modify the vascular effects occurring in hemorrhoid disease when it is used as an intra-anal ointment. Thereby decrease or eliminate the most frequently occurring symptoms of hemorrhoid disease[1]. |
| Alias | S-MPEC |
| Molecular Weight | 348.48 |
| Formula | C23H28N2O |
| Cas No. | 58754-46-4 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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