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Naloxegol oxalate
🥰Excellent
Catalog No. T3355Cas No. 1354744-91-4
Alias NKTR-118 oxalate, NKTR118 oxalate, AZ-13337019 oxalate, AZ 13337019 oxalate
Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
Naloxegol oxalate
🥰Excellent
Purity: 100%
Catalog No. T3355Alias NKTR-118 oxalate, NKTR118 oxalate, AZ-13337019 oxalate, AZ 13337019 oxalateCas No. 1354744-91-4
Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $40 | In Stock | |
| 10 mg | $56 | In Stock | |
| 25 mg | $92 | In Stock | |
| 50 mg | $133 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $66 | In Stock |
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Purity:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation. |
| Alias | NKTR-118 oxalate, NKTR118 oxalate, AZ-13337019 oxalate, AZ 13337019 oxalate |
| Molecular Weight | 741.83 |
| Formula | C36H55NO15 |
| Cas No. | 1354744-91-4 |
| Smiles | COCCOCCOCCOCCOCCOCCOCCO[C@H]1CC[C@]2([C@H]3Cc4c5[C@]2([C@H]1Oc5c(cc4)O)CCN3CC=C)O.C(=O)(C(=O)O)O |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (67.4 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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