Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Seclidemstat (SP-2577) is an effective LSD1 inhibitor, with a mean IC50 of 127 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 41.00 | |
10 mg | In stock | $ 66.00 | |
25 mg | In stock | $ 123.00 | |
50 mg | In stock | $ 197.00 | |
100 mg | In stock | $ 373.00 | |
200 mg | In stock | $ 556.00 | |
500 mg | In stock | $ 896.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 45.00 |
Description | Seclidemstat (SP-2577) is an effective LSD1 inhibitor, with a mean IC50 of 127 nM. |
Targets&IC50 | LSD1:127 nM |
In vivo | Interstitial MR lymphography with gadopentetate dimeglumine (Gd-DTPA) allows clear visualization of the lymphatic pathway in healthy mice, and no significant difference is found between the two agents. Their rapid kinetics limits the imaging timing window, however, facilitates repeated assessment in a single imaging session [1]. Direct visualization of spilled gastrointestinal gadopentetate dimeglumine helps discriminate ischemic from control rats in this model [2]. |
Synonyms | SP-2577 |
Molecular Weight | 450.94 |
Formula | C20H23ClN4O4S |
CAS No. | 1423715-37-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: < 0.1 mg/mL (insoluble)
DMSO: 100 mg/mL (221.76 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
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