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Luxdegalutamide
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Luxdegalutamide
Catalog No. T75129Cas No. 2750830-09-0
Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the wild-type androgen receptor AR, as well as AR LBD mutants including those associated with the most prevalent pathogenic AR L702H, H875Y and T878A mutations.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $318 | In Stock | |
| 5 mg | $768 | In Stock | |
| 10 mg | $1,180 | In Stock | |
| 25 mg | $1,780 | In Stock | |
| 50 mg | $2,320 | In Stock | |
| 100 mg | $2,970 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the wild-type androgen receptor AR, as well as AR LBD mutants including those associated with the most prevalent pathogenic AR L702H, H875Y and T878A mutations. |
| Alias | ARV-766 |
| Molecular Weight | 807.95 |
| Formula | C45H54FN7O6 |
| Cas No. | 2750830-09-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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