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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $71 | In Stock | |
5 mg | $178 | In Stock | |
10 mg | $238 | In Stock | |
25 mg | $397 | In Stock | |
50 mg | $567 | In Stock | |
100 mg | $768 | In Stock | |
500 mg | $1,540 | In Stock | |
1 mL x 10 mM (in DMSO) | $196 | In Stock |
Description | DBPR108 is an orally bioavailable dipeptide-derived DPP4 inhibitor (IC50: 15 nM) and it has no inhibition on DDP8 and DPP9. |
In vitro | DBPR108 displays a more than 3000-fold selectivity over DPP8 DPP9, FAP and DPP-II. |
In vivo | DBPR108 is a potent, selective, long-acting and safe DPP-IV inhibitor as a potential treatment of type 2 diabetes mellitus. The in vivo effects of DBPR108, including inhibition of plasma DPP-IV activity and suppression of blood glucose elevation, were also demonstrated. |
Molecular Weight | 324.39 |
Formula | C16H25FN4O2 |
Cas No. | 1186426-66-3 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||||||||||||
Solubility Information | DMSO: ≥ 25 mg/mL (77.07 mM) | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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