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Dibenamine hydrochloride
🥰Excellent
Catalog No. T37906Cas No. 55-43-6
Dibenamine hydrochloride is a competitive and irreversible blocker of the β-adrenergic receptor.
Dibenamine hydrochloride
🥰Excellent
Purity: 96.43%
Catalog No. T37906Cas No. 55-43-6
Dibenamine hydrochloride is a competitive and irreversible blocker of the β-adrenergic receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 500 mg | $29 | In Stock |
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Octopamine hydrochloride
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Trazodone hydrochloride
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Mianserin hydrochloride
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Dexmedetomidine hydrochloride
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Isoprenaline hydrochloride
Cited
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Purity:96.43%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Dibenamine hydrochloride is a competitive and irreversible blocker of the β-adrenergic receptor. |
| In vitro | The irreversible inhibitory effects of dibenamine on the noradrenaline-, K- and Ba-induced contractions of rat's isolated vas deferens, particularly in relation to Ca. |
| In vivo | Dibenamine hydrochloride causes a significant increase in the rate of destruction of L-epinephrine in the mouse. Pretreatment with Dibenamine hydrochloride apparently slowed the conversion of Ccl4 to CHCL3. Dibenamine hydrochloride (25 mg/kg; s.c.) decreased the CHCl3, levels at 2 and 6 hr by 30%-50%[3]. |
| Molecular Weight | 296.23 |
| Formula | C16H19Cl2N |
| Cas No. | 55-43-6 |
| Smiles | Cl.ClCCN(Cc1ccccc1)Cc1ccccc1 |
| Relative Density. | 1.107g/cm3 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 125 mg/mL (421.97 mM) H2O: 33.33 mg/mL (112.51 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
H2O/DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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