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Fadrozole hydrochloride
🥰Excellent
Catalog No. T7556Cas No. 102676-31-3
Alias CGS 16949A
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that effectively suppresses estrogen production in fish ovaries.
Fadrozole hydrochloride
🥰Excellent
Catalog No. T7556Alias CGS 16949ACas No. 102676-31-3
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that effectively suppresses estrogen production in fish ovaries.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $42 | In Stock | |
| 10 mg | $66 | In Stock | |
| 25 mg | $128 | In Stock | |
| 50 mg | $227 | In Stock | |
| 100 mg | $398 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $46 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that effectively suppresses estrogen production in fish ovaries. |
| Targets&IC50 | Aromatase:1.4 nM (rat), Aromatase:5 nM(human) |
| In vivo | Fadrozole hydrochloride inhibits growth of androstenedione-stimulated mammary D2 cells implanted into thoracic mammary fat pads of mice by 95% when administered at a dose of 0.5 mg per animal per day. |
| Alias | CGS 16949A |
| Molecular Weight | 259.73 |
| Formula | C14H14ClN3 |
| Cas No. | 102676-31-3 |
| Smiles | Cl.N#Cc1ccc(cc1)C1CCCc2cncn12 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 100 mg/mL (385.02 mM) H2O: 100 mg/mL (385.02 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO/H2O
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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