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Mocravimod hydrochloride
Catalog No. T12086Cas No. 509088-69-1
Mocravimod hydrochloride (KRP-203) is an effecitive and orally active agonist of sphingosine 1-phosphate receptor type 1(S1PR1).
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $64 | In Stock | |
| 5 mg | $172 | In Stock | |
| 10 mg | $278 | In Stock | |
| 25 mg | $563 | In Stock | |
| 50 mg | $872 | In Stock | |
| 100 mg | $1,170 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $182 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Mocravimod hydrochloride (KRP-203) is an effecitive and orally active agonist of sphingosine 1-phosphate receptor type 1(S1PR1). |
| In vivo | In mHC-disparate rat heart allografts, Mocravimod hydrochloride(orally; 0.1 and 1 mg/kg/day; for 100 days) prolongs graft survival and attenuates chronic rejection[1]. Mocravimod hydrochloride ameliorates atherosclerosis in LDL-R(-/-) Mice[2]. |
| Alias | KRP-203 |
| Molecular Weight | 480.45 |
| Formula | C24H27Cl2NO3S |
| Cas No. | 509088-69-1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 95 mg/mL (197.73 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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