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N-Methylcytisine

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Purity:99.83%

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COA HNMR HPLC

N-Methylcytisine

Catalog No. T5S0994Cas No. 486-86-2

1. N-Methylcytisine (Caulophylline)'s nicotinic receptors have high affinity (KD = 5 nM)to nAChR from squid optical ganglia. 2. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).

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Pack Size	Price	Availability
1 mg	$59	In Stock
5 mg	$129	In Stock
10 mg	$219	In Stock
25 mg	$389	In Stock
50 mg	$573	In Stock
100 mg	$835	In Stock
500 mg	$1,680	In Stock
1 mL x 10 mM (in DMSO)	$137	In Stock

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Product Introduction

Bioactivity

Description	1. N-Methylcytisine (Caulophylline)'s nicotinic receptors have high affinity (KD = 5 nM)to nAChR from squid optical ganglia. 2. N-Methylcytisine and N, N-dimethylcytisine did not displace 14C-tubocurarine at a concentration of .1 mM, cytisine was the only effective inhibitor of 14C-tubocurarine specific binding (Ki=7 nM).
Alias	Caulophylline

Chemical Properties

Molecular Weight	204.27
Formula	C12H16N2O
Cas No.	486-86-2

Storage & Solubility Information

Storage

keep away from direct sunlight Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 27.5 mg/mL (134.62 mM)

Chloroform, Dichloromethane, Ethyl Acetate, Acetone, etc.: Soluble

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	4.8955 mL	24.4774 mL	48.9548 mL	244.7741 mL
5 mM	0.9791 mL	4.8955 mL	9.7910 mL	48.9548 mL
10 mM	0.4895 mL	2.4477 mL	4.8955 mL	24.4774 mL
20 mM	0.2448 mL	1.2239 mL	2.4477 mL	12.2387 mL
50 mM	0.0979 mL	0.4895 mL	0.9791 mL	4.8955 mL
100 mM	0.0490 mL	0.2448 mL	0.4895 mL	2.4477 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Tech Support

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