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N6-Ethyladenosine
Catalog No. T12161Cas No. 14357-08-5
N6-Ethyladenosine, an adenosine derivative, acts as an agonist of Adenosine receptors (hA1AR and hA3AR) with Ki values of 4.9 nM and 4.7 nM, respectively.
N6-Ethyladenosine
Catalog No. T12161Cas No. 14357-08-5
N6-Ethyladenosine, an adenosine derivative, acts as an agonist of Adenosine receptors (hA1AR and hA3AR) with Ki values of 4.9 nM and 4.7 nM, respectively.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $29 | In Stock | |
| 5 mg | $46 | In Stock | |
| 10 mg | $73 | In Stock | |
| 25 mg | $133 | In Stock | |
| 50 mg | $223 | In Stock | |
| 100 mg | $329 | In Stock | |
| 200 mg | $475 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $78 | In Stock |
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CitedSelect Batch
Purity:99.96%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | N6-Ethyladenosine, an adenosine derivative, acts as an agonist of Adenosine receptors (hA1AR and hA3AR) with Ki values of 4.9 nM and 4.7 nM, respectively. |
| Targets&IC50 | A3AR (human):4.7 nM (ki), A1AR (human):4.9 nM (Ki) |
| In vitro | N6-Ethyladenosine exhibits more selectivity at hA1AR and hA3AR over hA2AR with Ki of 8900±770 nM [1]. |
| Molecular Weight | 295.29 |
| Formula | C12H17N5O4 |
| Cas No. | 14357-08-5 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 83.33 mg/mL (282.20 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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