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NS-2710
Catalog No. T28197Cas No. 184220-36-8
Alias NS2710, NS 2710
NS-2710 is a non-selective GABA(A) receptor partial agonist for the study of anxiety disorders.
NS-2710
Purity: 99.82%
Catalog No. T28197Alias NS2710, NS 2710Cas No. 184220-36-8
NS-2710 is a non-selective GABA(A) receptor partial agonist for the study of anxiety disorders.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $293 | In Stock | |
| 5 mg | $722 | In Stock | |
| 10 mg | $987 | In Stock | |
| 25 mg | $1,520 | In Stock | |
| 50 mg | $1,980 | In Stock |
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Purity:99.82%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | NS-2710 is a non-selective GABA(A) receptor partial agonist for the study of anxiety disorders. |
| In vivo | NS2710 was administered orally to mice 15 minutes prior to testing at doses of 1.0, 3.0, and 10.0 mg/kg. NS2710 at doses of 3.0 and 10.0 mg/kg increased response rates, independent of baseline response rates and whether responses were penalized. When differentiating between baseline rates, the effect of composition was highly significant [F(1,7) = 38.9, P < 0.001], and the interaction between composition and treatment was not significant, but the main effect of treatment was significant [F(3,21) = 5.0, P < 0.01]. In both cases, post hoc tests showed that NS2710 at doses of 3.0 and 10.0 mg/kg increased response rates regardless of whether response was penalized or unpunished [2]. |
| Alias | NS2710, NS 2710 |
| Molecular Weight | 356.42 |
| Formula | C22H20N4O |
| Cas No. | 184220-36-8 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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