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Ralfinamide
Catalog No. T7349Cas No. 133865-88-0
Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $45 | In Stock | |
| 10 mg | $72 | In Stock | |
| 25 mg | $148 | In Stock | |
| 50 mg | $275 | In Stock | |
| 100 mg | $419 | In Stock | |
| 200 mg | $619 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $79 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions. |
| In vivo | Oral ralfinamide dose-dependently alleviated spared nerve injury-induced allodynia in rats and mice. Ralfinamide increased mechanical withdrawal thresholds in oxaliplatin-induced and paclitaxel-induced neuropathic pain. Ralfinamide did not affect physiological pain, locomotion,or cardiovascular function[1]. |
| Alias | Priralfinamide, FCE-26742A |
| Molecular Weight | 302.34 |
| Formula | C17H19FN2O2 |
| Cas No. | 133865-88-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 125 mg/mL (413.44 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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