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(Rac)-VU 6008667
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(Rac)-VU 6008667
Catalog No. T12679Cas No. 2092917-63-8
(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) with IC50 of 1.8 μM and pIC50 of 5.75, has high CNS penetration.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $54 | In Stock | |
| 5 mg | $148 | In Stock | |
| 10 mg | $273 | In Stock | |
| 25 mg | $459 | In Stock | |
| 50 mg | $677 | In Stock | |
| 100 mg | $963 | In Stock | |
| 500 mg | $1,930 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | (Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) with IC50 of 1.8 μM and pIC50 of 5.75, has high CNS penetration. |
| Molecular Weight | 438.85 |
| Formula | C24H17ClF2N2O2 |
| Cas No. | 2092917-63-8 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||
| Solubility Information | DMSO: 20 mg/mL (45.57 mM)  H2O: 0.1 mg/mL (insoluble) | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
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