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3-Bromocytisine

🥰Excellent
Catalog No. T10108Cas No. 207390-14-5
Alias 3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-Bromocytisine

3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).

3-Bromocytisine

3-Bromocytisine

🥰Excellent
Purity: 98.14%
Catalog No. T10108Alias 3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-BromocytisineCas No. 207390-14-5
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
Pack SizePriceAvailabilityQuantity
1 mg91 €In Stock
5 mg227 €In Stock
10 mg308 €In Stock
25 mg520 €In Stock
50 mg748 €In Stock
100 mg1.026 €In Stock
1 mL x 10 mM (in DMSO)208 €In Stock
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Purity:98.14%
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Product Introduction

Bioactivity
Description
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
Targets&IC50
α4β4 (human):0.28 nM , α4β2 (human):0.30 nM , α7 (human):31.6 nM
In vitro
3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively [2].
Alias3-Br-cytisine, (-)-9-Bromocytisine, (-)-3-Bromocytisine
Chemical Properties
Molecular Weight269.14
FormulaC11H13BrN2O
Cas No.207390-14-5
SmilesO=C1N2C([C@@]3(C[C@](C2)(CNC3)[H])[H])=CC=C1Br
Relative Density.1.61 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 50 mg/mL (185.78 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.7155 mL18.5777 mL37.1554 mL185.7769 mL
5 mM0.7431 mL3.7155 mL7.4311 mL37.1554 mL
10 mM0.3716 mL1.8578 mL3.7155 mL18.5777 mL
20 mM0.1858 mL0.9289 mL1.8578 mL9.2888 mL
50 mM0.0743 mL0.3716 mL0.7431 mL3.7155 mL
100 mM0.0372 mL0.1858 mL0.3716 mL1.8578 mL

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