Powder: -20°C for 3 years | In solvent: -80°C for 1 year
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 96.00 | |
5 mg | In stock | $ 239.00 | |
10 mg | In stock | $ 325.00 | |
25 mg | In stock | $ 548.00 | |
50 mg | In stock | $ 788.00 | |
100 mg | In stock | $ 1,080.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 219.00 |
Description | 3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7). |
Targets&IC50 | α4β4 (human):0.28 nM , α7 (human):31.6 nM , α4β2 (human):0.30 nM |
In vitro | 3-Bromocytisine shows different effects on high and low ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively [2]. |
Synonyms | (-)-3-Bromocytisine, (-)-9-Bromocytisine, 3-Br-cytisine |
Molecular Weight | 269.14 |
Formula | C11H13BrN2O |
CAS No. | 207390-14-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (185.78 mM)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
3-Bromocytisine 207390-14-5 Neuroscience AChR (-)-3-Bromocytisine (-)-9-Bromocytisine 3-Br-cytisine 9-Bromocytisine inhibitor inhibit