Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AC-55541 (AOB2796) is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays, with potencies ranging from 200 to 1000 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 36.00 | |
5 mg | In stock | $ 85.00 | |
10 mg | In stock | $ 148.00 | |
25 mg | In stock | $ 253.00 | |
50 mg | In stock | $ 377.00 | |
100 mg | In stock | $ 558.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 97.00 |
Description | AC-55541 (AOB2796) is a novel PAR2 agonist; activated PAR2 signaling in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays, with potencies ranging from 200 to 1000 nM. |
Targets&IC50 | PAR2:200-1000 nM(EC50) |
Kinase Assay | Inhibition Kinetics Studies: Recombinant human wild-type and T790M/L858R double mutant EGFR, both Nterminal GST-tagged, are used in the assay. The Omnia continuous read assay is performed as described by the vendor. |
Synonyms | AOB2796 |
Molecular Weight | 518.36 |
Formula | C25H20BrN5O3 |
CAS No. | 916170-19-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 5.18 mg/mL (10 mM), Sonification is recommended
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
AC-55541 916170-19-9 GPCR/G Protein Proteases/Proteasome Ubiquitination Protease-activated Receptor Proteasome inhibit AC 55541 AOB-2796 Inhibitor Protease Activated Receptor (PAR) AOB 2796 Thrombin receptors AOB2796 AC55541 inhibitor