Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 38.00 | |
5 mg | In stock | $ 89.00 | |
10 mg | In stock | $ 155.00 | |
25 mg | In stock | $ 312.00 | |
50 mg | In stock | $ 588.00 | |
100 mg | In stock | $ 843.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 98.00 |
Description | Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM). |
Targets&IC50 | CYP2D6:5.4 μM |
In vitro | Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively[1]. |
Molecular Weight | 389.47 |
Formula | C23H24FN5 |
CAS No. | 1186430-60-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 11 mg/mL (28.24 mM)
You can also refer to dose conversion for different animals. More
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Antihistamine-1 1186430-60-3 Metabolism P450 Antihistamine1 Antihistamine 1 inhibitor inhibit