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Gluten Exorphin C
🥰Excellent
Catalog No. TP1832Cas No. 142479-62-7
Gluten exorphin C is an opioid peptide derived from wheat gluten, with IC50 values of 40 μM for μ opioid and 13.5 μM for δ opioid activities in the GPI and MVD assays, respectively. Isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten, it is considered a δ-opioid receptor-selective ligand.
Gluten Exorphin C
🥰Excellent
Purity: 100%
Catalog No. TP1832Cas No. 142479-62-7
Gluten exorphin C is an opioid peptide derived from wheat gluten, with IC50 values of 40 μM for μ opioid and 13.5 μM for δ opioid activities in the GPI and MVD assays, respectively. Isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten, it is considered a δ-opioid receptor-selective ligand.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $39 | In Stock | |
| 5 mg | $97 | In Stock | |
| 10 mg | $147 | In Stock | |
| 25 mg | $248 | In Stock | |
| 50 mg | $369 | In Stock | |
| 100 mg | $543 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Gluten exorphin C is an opioid peptide derived from wheat gluten, with IC50 values of 40 μM for μ opioid and 13.5 μM for δ opioid activities in the GPI and MVD assays, respectively. Isolated from the pepsin-trypsin-chymotrypsin digest of wheat gluten, it is considered a δ-opioid receptor-selective ligand. |
| Targets&IC50 | δ opioid:13.5 μM (IC50), μ opioid:40 μM (IC50) |
| Molecular Weight | 591.7 |
| Formula | C29H45N5O8 |
| Cas No. | 142479-62-7 |
| Smiles | CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(O)=O |
| Relative Density. | 1.264 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 10 mM | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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