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Mirogabalin
🥰Excellent
Catalog No. T7216Cas No. 1138245-13-2
Alias DS5565
Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.
Mirogabalin
🥰Excellent
Purity: 99.89%
Catalog No. T7216Alias DS5565Cas No. 1138245-13-2
Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $35 | In Stock | |
| 5 mg | $81 | In Stock | |
| 10 mg | $127 | In Stock | |
| 25 mg | $222 | In Stock | |
| 50 mg | $338 | In Stock | |
| 100 mg | $513 | In Stock | |
| 500 mg | $1,080 | In Stock |
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Purity:99.89%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects. |
| In vivo | Mirogabalin has potent and sustained analgesic effects (ED50 = 2.5 mg/kg) in rats with diabetes induced by streptozotocin .?Mirogabalin does not inhibit activities associated with CNS adverse effects of analgesics, such as rotarod performance (ID50 = 9.4 mg/kg) or locomotor activity (ID50 = 43.9 mg/kg), at its effective dose. |
| Alias | DS5565 |
| Molecular Weight | 209.28 |
| Formula | C12H19NO2 |
| Cas No. | 1138245-13-2 |
| Smiles | CCC1=C[C@@H]2[C@@H](C[C@]2(CN)CC(O)=O)C1 |
| Relative Density. | 1.104 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||
| Solubility Information | DMSO: 1.83 mg/mL (8.76 mM), Sonication is recommended.  | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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