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[11C]MP 10
![[11C]MP 10](/group3/M00/03/29/CgoaEGY7SLaEXVj0AAAAAK5zpaY421.png)
[11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.
Catalog No. T6042Cas No. 1292799-56-4
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Purity:99.87%
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[11C]MP 10
Catalog No. T6042Alias PF-2545920, MardepodectCas No. 1292799-56-4
[11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $55 | In Stock | |
| 2 mg | $98 | In Stock | |
| 5 mg | $202 | In Stock | |
| 10 mg | $279 | In Stock | |
| 25 mg | $455 | In Stock | |
| 50 mg | $669 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $216 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
| Description | [11C]MP 10 (PF-2545920), a specific and effective PDE10A inhibitor (IC50=0.37 nM), is with more than1000-fold specificity activity over the PDE. |
| Targets&IC50 | PDE10A:0.37 nM |
| In vitro | PF-2545920 shows excellent potency and specificity in PDE10A with IC50 of 1.26 nM. |
| Alias | PF-2545920, Mardepodect |
| Molecular Weight | 391.45 |
| Formula | C25H20N4O |
| Cas No. | 1292799-56-4 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| Solubility Information | Ethanol: 69 mg/mL (175.8 mM) DMSO: 79 mg/mL (201.29 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
Ethanol/DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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