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Azimilide Dihydrochloride
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Azimilide Dihydrochloride
Catalog No. T7505Cas No. 149888-94-8
Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the slowly activating (IKs) and rapidly activating (IKr) components of the delayed rectifier potassium current
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $43 | In Stock | |
| 10 mg | $61 | In Stock | |
| 25 mg | $136 | In Stock | |
| 50 mg | $263 | In Stock | |
| 100 mg | $498 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $51 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the slowly activating (IKs) and rapidly activating (IKr) components of the delayed rectifier potassium current |
| In vivo | Azimilide has shown excellent efficacy (>85%) in suppressing supraventricular arrhythmias in a variety of dog models.?It also suppressed complex ventricular arrhythmias in infarcted dogs and, in a sudden death cardiac model, decreased mortality[1]. |
| Alias | NE-10064 Dihydrochloride |
| Molecular Weight | 530.88 |
| Formula | C23H30Cl3N5O3 |
| Cas No. | 149888-94-8 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||
| Solubility Information | DMSO: 8.46 mg/mL (15.94 mM) | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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