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BMS-929075
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BMS-929075
Catalog No. T26863Cas No. 1217338-97-0
BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic parameters.BMS-929075 shows cytotoxicity.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $190 | In Stock | |
| 5 mg | $480 | In Stock | |
| 10 mg | $687 | In Stock | |
| 25 mg | $1,080 | In Stock | |
| 50 mg | $1,480 | In Stock | |
| 100 mg | $1,990 | In Stock | |
| 500 mg | $3,920 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $598 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic parameters.BMS-929075 shows cytotoxicity. |
| In vitro | BMS-929075 (0-60 µM) showed cytotoxicity with CC50 values of 60, >12.5, and >50 µM for Huh-7, HepG2, and primary human hepatocytes, respectively.[1] |
| In vivo | BMS-929075 (i.v. 2 mg/kg; orally 6 mg/kg) showed good pharmacokinetic parameters with an oral bioavailability of 48% in rats.[1] |
| Alias | BMS 929075, BMS929075 |
| Molecular Weight | 538.54 |
| Formula | C31H24F2N4O3 |
| Cas No. | 1217338-97-0 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 27.5 mg/mL (51.06 mM)  | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
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