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Diminazene is a trypanocidal agent.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
100 mg | 39 € | In Stock |
Description | Diminazene is a trypanocidal agent. |
In vitro | Administering 7 mg/kg, i.m. of Diminazene aceturate effectively clears parasites from the bloodstream of infected dogs. An initial treatment dose of 3.5 mg/kg of Diminazene aceturate significantly alleviates T. evansi infection in horses and mules, with parasites being eliminated from the peripheral blood within 1-7 days and 1-14 days, respectively. |
In vivo | Transport of [3H] diminazene is substantially inhibited by pentamidine and adenosine, with Ki values of 0.21 μM and 0.25 μM, respectively. Notably, [3H] diminazene accumulates in yeast cells expressing TbAT1 at a rate of 0.0083 pmol/10^7 cells/s when treated with 2.5 μM of the radioactive compound, and this accumulation is completely suppressed by 1 mM of unlabeled Diminazene Aceturate. |
Alias | DIZE |
Molecular Weight | 515.52 |
Formula | C22H29N9O6 |
Cas No. | 908-54-3 |
Smiles | c1(ccc(cc1)/N=N/Nc1ccc(cc1)C(=N)N)C(=N)N.CC(=O)NCC(=O)O.CC(=O)NCC(=O)O |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | H2O: 92 mg/mL (178.5 mM) Ethanol: < 1 mg/mL (insoluble or slightly soluble) DMSO: 1 mg/mL, Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
H2O
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