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Ezatiostat TFA
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Ezatiostat TFA
Catalog No. T5862
Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $50 | In Stock | |
| 5 mg | $60 | In Stock | |
| 10 mg | $102 | In Stock | |
| 25 mg | $233 | In Stock | |
| 50 mg | $308 | In Stock | |
| 100 mg | $477 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $116 | In Stock |
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CitedProduct Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Ezatiostat TFA (TLK199) is a liposomal small-molecule glutathione analog inhibitor of glutathione S-transferase (GST) P1-1 with hematopoiesis-stimulating activity. |
| In vitro | Ezatiostat is a tripeptide analog of glutathione that can selectively inhibit GSTP1-1 catalytic activity (Ki = 400 nM) with minimal effect on the related GSTα and -μ families (Kis range from 20-75 μM)[1]. |
| Alias | TER199(free base), Ezatiostat TFA (free base), Ezatiostat, TLK199 |
| Molecular Weight | 643.67 |
| Formula | C29H36F3N3O8S |
| Cas No. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||
| Solubility Information | DMSO: 25 mg/mL (47.2 mM)  | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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