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GSK3787

🥰Excellent
Catalog No. T1941Cas No. 188591-46-0

GSK3787 is a specific and irreversible PPARδ inhibitor(pIC50= 6.6).

GSK3787

GSK3787

🥰Excellent
Purity: 98.53%
Catalog No. T1941Cas No. 188591-46-0
GSK3787 is a specific and irreversible PPARδ inhibitor(pIC50= 6.6).
Pack SizePriceAvailabilityQuantity
5 mg$50In Stock
10 mg$79In Stock
25 mg$183In Stock
50 mg$325In Stock
100 mg$548In Stock
500 mg$1,170In Stock
1 mL x 10 mM (in DMSO)$50In Stock
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Purity:98.53%
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Product Introduction

Bioactivity
Description
GSK3787 is a specific and irreversible PPARδ inhibitor(pIC50= 6.6).
Targets&IC50
PPARδ:6.6(pIC50)
In vivo
Pparβ/δ-null mice are administered GSK3787 (10 mg/kg) by oral gavage 3 hours before euthanasia.
Chemical Properties
Molecular Weight392.78
FormulaC15H12ClF3N2O3S
Cas No.188591-46-0
SmilesFC(F)(F)c1ccc(nc1)S(=O)(=O)CCNC(=O)c1ccc(Cl)cc1
Relative Density.1.448 g/cm3 at 20℃
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: 40 mg/mL (101.84 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.5460 mL12.7298 mL25.4595 mL127.2977 mL
5 mM0.5092 mL2.5460 mL5.0919 mL25.4595 mL
10 mM0.2546 mL1.2730 mL2.5460 mL12.7298 mL
20 mM0.1273 mL0.6365 mL1.2730 mL6.3649 mL
50 mM0.0509 mL0.2546 mL0.5092 mL2.5460 mL
100 mM0.0255 mL0.1273 mL0.2546 mL1.2730 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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