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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $155 | In Stock | |
5 mg | $328 | In Stock | |
10 mg | $563 | In Stock | |
25 mg | $890 | In Stock | |
50 mg | $1,230 | In Stock | |
100 mg | $1,670 | In Stock | |
1 mL x 10 mM (in DMSO) | $363 | In Stock |
Description | Nampt-IN-5 is a potent and orally active inhibitor of nicotinamide phosphoribosyltransferase (NAMPT) . |
In vitro | Nampt-IN-5 shows a good ADME data: mouse microsomal clearance, CYP3A4 inhibition value (0.75 μM), Sol6.8: 0.056 mM; MDCK Papp AB: 18.6.Nampt-IN-5 has cellular IC50s of 0.7 nM and 3.9 nM against A2780 and COR-L23, respectively in CellTiterGlo (CTG) assays[1]. |
Molecular Weight | 427.5 |
Formula | C25H25N5O2 |
Cas No. | 2380013-17-0 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 48 mg/mL (112.28 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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