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Nerisopam
🥰Excellent
Catalog No. T28159Cas No. 102771-12-0
Alias GYKI-52322, GYKI52322, GYKI 52322, EGIS-6775, EGIS6775
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
Nerisopam
🥰Excellent
Purity: 97.27%
Catalog No. T28159Alias GYKI-52322, GYKI52322, GYKI 52322, EGIS-6775, EGIS6775Cas No. 102771-12-0
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $142 | In Stock | |
| 5 mg | $350 | In Stock | |
| 10 mg | $530 | In Stock | |
| 25 mg | $859 | In Stock | |
| 50 mg | $1,180 | In Stock | |
| 100 mg | $1,590 | In Stock | |
| 500 mg | $3,190 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $475 | In Stock |
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CitedSelect Batch
Purity:97.27%
Contact us for more batch information
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor. |
| In vivo | Nerisopam application (30 mg/kg; 5 h; gastric cannula) cells in the reticular zone of the substantia nigra showed Fos-like immunopositivity.[6] Nerisopam (20 mg/kg;13 days; daily) for two weeks after a daily application, relatively weak Fos-like immunoreactivity was observed in the striatum and the subthalamic nucleus but not in the globus pallidus. Our results suggest that the striatal neurons are the primary targets of this anxiolytic and antipsychotic drug in the central nervous system.[6] |
| Alias | GYKI-52322, GYKI52322, GYKI 52322, EGIS-6775, EGIS6775 |
| Molecular Weight | 309.36 |
| Formula | C18H19N3O2 |
| Cas No. | 102771-12-0 |
| Smiles | O(C)C=1C=C2C(=NN=C(C)CC2=CC1OC)C3=CC=C(N)C=C3 |
| Relative Density. | 1.22 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 25 mg/mL (41.38 mM)  | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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