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YYA-021
Catalog No. T6256Cas No. 144217-65-2
Alias YYA 021
YYA-021 inhibits HIV entry, with high anti-HIV activity and low cytotoxicity.
YYA-021
Catalog No. T6256Alias YYA 021Cas No. 144217-65-2
YYA-021 inhibits HIV entry, with high anti-HIV activity and low cytotoxicity.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 5 mg | $35 | In Stock | |
| 10 mg | $43 | In Stock | |
| 25 mg | $93 | In Stock | |
| 50 mg | $129 | In Stock | |
| 100 mg | $167 | In Stock | |
| 200 mg | $247 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $39 | In Stock |
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CitedSelect Batch
Purity:100%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | YYA-021 inhibits HIV entry, with high anti-HIV activity and low cytotoxicity. |
| Targets&IC50 | HIV:8.4 μM |
| In vitro | YYA-021 enhances the neutralization sensitivity of simian-human immunodeficiency virus (SHIV) carrying the envelope from the clade B clinical human immunodeficiency virus type 1 (HIV-1) isolate MNA. [1] |
| In vivo | In rats and rhesus macaques, YYA-021 (i.v.) shows moderate half-lives, wide tissue distribution and relatively high distribution volumes. [2] |
| Alias | YYA 021 |
| Molecular Weight | 317.43 |
| Formula | C18H27N3O2 |
| Cas No. | 144217-65-2 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 11 mg/mL (34.65 mM), Sonication is recommended.  H2O: < 0.1 mg/mL (insoluble) | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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