Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 64.00 | |
10 mg | In stock | $ 106.00 | |
25 mg | In stock | $ 219.00 | |
50 mg | In stock | $ 396.00 | |
100 mg | In stock | $ 595.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 70.00 |
Description | AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration. |
Targets&IC50 | δ opioid receptor: |
In vitro | Does not trigger acute desensitization of the analgesic response |
In vivo | Reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration. |
Synonyms | ARM390 Hydrochloride, ARM-390 HCl |
Molecular Weight | 384.94 |
Formula | C23H29ClN2O |
CAS No. | 209808-47-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: 38.49 mg/mL (100 mM)
DMSO: 38.49 mg/mL (100 mM)
You can also refer to dose conversion for different animals. More
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