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BTRX-335140
Contact us for more batch information
BTRX-335140
Catalog No. T14835Cas No. 2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. BTRX-335140 can distribute well into the CNS. ADMET (absorption, distribution, metabolism, excretion, and toxicity) . BTRX-335140 endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $107 | In Stock | |
| 2 mg | $157 | In Stock | |
| 5 mg | $263 | In Stock | |
| 10 mg | $428 | In Stock | |
| 25 mg | $885 | In Stock | |
| 50 mg | $1,450 | In Stock | |
| 100 mg | $1,980 | In Stock | |
| 200 mg | $2,770 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $297 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 values of 0.8 nM, 110 nM, and 6500 nM, respectively. BTRX-335140 can distribute well into the CNS. ADMET (absorption, distribution, metabolism, excretion, and toxicity) . BTRX-335140 endows with favorable in vitro ADMET and in vivo pharmacokinetic profiles and medication-like duration of action in rats. |
| Alias | CYM-53093 |
| Molecular Weight | 453.55 |
| Formula | C25H32FN5O2 |
| Cas No. | 2244614-14-8 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | ||||||||||||||||||||
| Solubility Information | DMSO: 5.5 mg/mL (12.13 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
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