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CEP-37440 is an effective and specific Dual FAK/ALK inhibitor with IC50s of 120 nM(ALK cellular in 75% human plasma) and 2.3 nM (FAK).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $31 | In Stock | |
2 mg | $44 | In Stock | |
5 mg | $72 | In Stock | |
10 mg | $128 | In Stock | |
25 mg | $269 | In Stock | |
50 mg | $513 | In Stock | |
100 mg | $746 | In Stock |
Description | CEP-37440 is an effective and specific Dual FAK/ALK inhibitor with IC50s of 120 nM(ALK cellular in 75% human plasma) and 2.3 nM (FAK). |
Targets&IC50 | FAK:2.3 nM, ALK:120 nM |
Kinase Assay | Kinase assay: Inhibitory potency of GSK2656157 is measured using recombinant GST-PERK (536–1116 amino acids) with 6-His-full-length human eIF2a as a substrate. Kinase selectivity is evaluated using 27 kinases at GSK as well as a panel of 300 kinases. |
Alias | CEP37440 |
Molecular Weight | 580.12 |
Formula | C30H38ClN7O3 |
Cas No. | 1391712-60-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||
Solubility Information | DMSO: 2.2 mg/mL (3.79 mM), Sonication is recommended. | ||||||||||
Solution Preparation Table | |||||||||||
DMSO
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