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Vilaprisan
🥰Excellent
Catalog No. T35054Cas No. 1262108-14-4
Alias BAY10-02670, BAY-10-02670, BAY-1002670, BAY1002670, BAY 10-02670, BAY 1002670
Vilaprisan (BAY 1002670) is a novel orally available and selective progesterone receptor modulator (SPRM) with antiproliferative activity against uterine fibroids (UF) and can be used for the study of uterine fibroids.
Vilaprisan
🥰Excellent
Purity: 100%
Catalog No. T35054Alias BAY10-02670, BAY-10-02670, BAY-1002670, BAY1002670, BAY 10-02670, BAY 1002670Cas No. 1262108-14-4
Vilaprisan (BAY 1002670) is a novel orally available and selective progesterone receptor modulator (SPRM) with antiproliferative activity against uterine fibroids (UF) and can be used for the study of uterine fibroids.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | 185 € | In Stock | |
| 5 mg | 441 € | In Stock | |
| 10 mg | 645 € | In Stock | |
| 25 mg | 1.016 € | In Stock | |
| 50 mg | 1.358 € | In Stock | |
| 100 mg | 1.833 € | In Stock |
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Purity:100%
ee:97.88%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Vilaprisan (BAY 1002670) is a novel orally available and selective progesterone receptor modulator (SPRM) with antiproliferative activity against uterine fibroids (UF) and can be used for the study of uterine fibroids. |
| In vitro | Vilaprisan shows an IC50 of 0.09 nM in the PR transactivation assay[2]. |
| Alias | BAY10-02670, BAY-10-02670, BAY-1002670, BAY1002670, BAY 10-02670, BAY 1002670 |
| Molecular Weight | 544.57 |
| Formula | C27H29F5O4S |
| Cas No. | 1262108-14-4 |
| Smiles | C[C@@]12[C@]([C@]3(C([C@H](C1)C4=CC=C(S(C)(=O)=O)C=C4)=C5C(CC3)=CC(=O)CC5)[H])(CC[C@]2(C(C(F)(F)F)(F)F)O)[H] |
| Relative Density. | 1.41 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 7.86 mg/mL (14.43 mM)  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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