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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $122 | In Stock | |
5 mg | $297 | In Stock | |
10 mg | $463 | In Stock | |
25 mg | $766 | In Stock | |
50 mg | $1,070 | In Stock | |
100 mg | $1,450 | In Stock | |
1 mL x 10 mM (in DMSO) | $282 | In Stock |
Description | Furafylline is a selective inhibitor of human cytochrome P450 (CYP)1A2 (IC50 : 0.07 µM), |
Targets&IC50 | CYP1A2 (human):0.07 µM |
In vitro | Furafylline was a potent, non-competitive inhibitor of high affinity phenacetin O-deethylase activity of microsomal fractions of human liver, a reaction catalysed by P450IA2, with an IC50 value of 0.07 microM[1]. |
In vivo | Furafylline was originally introduced as a bronchodilator with extended duration compared to theophylline[1]. |
Molecular Weight | 260.25 |
Formula | C12H12N4O3 |
Cas No. | 80288-49-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
Solubility Information | DMSO: 12.5 mg/mL (48.03 mM) | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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