Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty

Methylnaltrexone bromide

🥰Excellent
Catalog No. T21422Cas No. 73232-52-7
Alias Relistor, MOA-728, MOA728, MOA 728, Methylnaltrexone

Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.

Methylnaltrexone bromide

Methylnaltrexone bromide

🥰Excellent
Purity: 99.02%
Catalog No. T21422Alias Relistor, MOA-728, MOA728, MOA 728, MethylnaltrexoneCas No. 73232-52-7
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.
Pack SizePriceAvailabilityQuantity
2 mg$47In Stock
5 mg$77In Stock
10 mg$118In Stock
25 mg$200In Stock
50 mg$286In Stock
100 mg$497In Stock
1 mL x 10 mM (in DMSO)$91In Stock
Bulk & Custom
Add to Cart
Questions
View More

Related Compound Libraries of "Methylnaltrexone bromide"

Select Batch
Purity:99.02%
Contact us for more batch information
Resource Download
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity
Description
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the side effects of opioid drugs such as constipation without affecting analgesia or precipitating withdrawals.
AliasRelistor, MOA-728, MOA728, MOA 728, Methylnaltrexone
Chemical Properties
Molecular Weight436.35
FormulaC21H26BrNO4
Cas No.73232-52-7
SmilesO=C1[C@@](OC2=C(O)C=CC3=C24)([H])[C@@]54CC[N+](C)(CC6CC6)[C@@](C3)([H])[C@]5(O)CC1.[Br-]
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
H2O: Insoluble
DMSO: 60 mg/ml (137.5 mM)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2917 mL11.4587 mL22.9174 mL114.5869 mL
5 mM0.4583 mL2.2917 mL4.5835 mL22.9174 mL
10 mM0.2292 mL1.1459 mL2.2917 mL11.4587 mL
20 mM0.1146 mL0.5729 mL1.1459 mL5.7293 mL
50 mM0.0458 mL0.2292 mL0.4583 mL2.2917 mL
100 mM0.0229 mL0.1146 mL0.2292 mL1.1459 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
%Tween 80
%ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy Methylnaltrexone bromide | purchase Methylnaltrexone bromide | Methylnaltrexone bromide cost | order Methylnaltrexone bromide | Methylnaltrexone bromide chemical structure | Methylnaltrexone bromide formula | Methylnaltrexone bromide molecular weight