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Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | 28 € | In Stock | |
10 mg | 45 € | In Stock | |
25 mg | 93 € | In Stock | |
50 mg | 150 € | In Stock | |
100 mg | 235 € | In Stock | |
200 mg | 335 € | In Stock | |
1 mL x 10 mM (in DMSO) | 29 € | In Stock |
Description | Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor. |
In vivo | Progabide ( 50, 100 and 200 mg/kg) given IP to male Wistar rats enhance the plasma corticosterone levels by 244, 365, and 476% respectively (t=6.44 to12.55, p<0.01). Progabide (10 mg/kg) fails to change the concentration of corticosterone in plasma (t=0.76, N.S.). The increased plasma corticosterone level induced by administration of 200 mg/kg Progabide is evident 30 (t=2.625, p<0.05), 60 (t=13.13, p<0.001) and 120 min (t=4.07, p<0.01) after drug injection, but returns to the control value 240 min after drug injection (t=0.86, N.S.). Compare with the corresponding control, The greatest corticosterone rise is reached 60 min following the administration of Progabide[1]. |
Alias | SL 76002, Halogabide, Gabrene, Gabren |
Molecular Weight | 334.77 |
Formula | C17H16ClFN2O2 |
Cas No. | 62666-20-0 |
Smiles | NC(=O)CCC\N=C(\c1ccc(Cl)cc1)c1cc(F)ccc1O |
Relative Density. | 1.2822 g/cm3 (Estimated) |
Storage | keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 225 mg/mL (672.1 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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