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(Rac)-Sabcomeline HCl
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(Rac)-Sabcomeline HCl
Catalog No. T68135LCas No. 133642-67-8
Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose. | Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $195 | In Stock | |
| 5 mg | $430 | In Stock | |
| 10 mg | $636 | In Stock | |
| 25 mg | $987 | In Stock | |
| 50 mg | $1,360 | In Stock | |
| 100 mg | $1,830 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Sabcomeline HCl is an M1 receptor agonist that can be used to study Alzheimer's disease. |
| In vivo | Sabcomeline HCl dose-dependently increased dopamine efflux in the medial prefrontal cortex but only a high dose of sabcomeline HCl (1 mg/kg; s.c.; rats) increased that in the nucleus accumbens. According to the analysis of net-AUC (area under the curve) values of acetylcholine and dopamine levels, the rank order of ability of these drugs to increase acetylcholine or dopamine levels is sabcomeline HCl>xanomeline approximately AC260584>N-desmethylclozapine.[5] |
| Alias | sabcomeline HCl(149156-36-5 Free base) |
| Molecular Weight | 229.71 |
| Formula | C10H16ClN3O |
| Cas No. | 133642-67-8 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (217.67 mM)  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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