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Tripelennamine hydrochloride
Catalog No. T1269Cas No. 154-69-8
Alias Tripelennamine HCl, Pyribenzamine hydrochloride, Pyribenzamine HCl
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
Tripelennamine hydrochloride
Catalog No. T1269Alias Tripelennamine HCl, Pyribenzamine hydrochloride, Pyribenzamine HClCas No. 154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 100 mg | $31 | In Stock | |
| 500 mg | $98 | In Stock | |
| 1 g | $142 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $30 | In Stock |
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation. |
| Targets&IC50 | H1 receptor:30 μM |
| In vitro | In equines, intravenous administration of Tripelennamine HCl (0.5 mg/kg) significantly elevates standing mixed venous blood oxygen tension and hemoglobin-O2 saturation while increasing oxygen content in both arterial and mixed venous blood, leading to central nervous system stimulation, resulting in heightened alertness and anxiety. |
| In vivo | In both human and rabbit liver microsomes, Tripelennamine inhibits the glucuronidation of 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine (PhIP). |
| Alias | Tripelennamine HCl, Pyribenzamine hydrochloride, Pyribenzamine HCl |
| Molecular Weight | 291.82 |
| Formula | C16H21N3·HCl |
| Cas No. | 154-69-8 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 13 mg/mL (44.55 mM)  | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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