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Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | 51 € | In Stock | |
2 mg | 74 € | In Stock | |
5 mg | 121 € | In Stock | |
10 mg | 169 € | In Stock | |
25 mg | 376 € | In Stock | |
50 mg | 559 € | In Stock | |
100 mg | 800 € | In Stock | |
1 mL x 10 mM (in DMSO) | 166 € | In Stock |
Description | Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM). |
Targets&IC50 | GR:0.9 nM (IC50) |
In vitro | AZD7594 shows no effect on progesterone receptor, mineralocorticoid receptor, Androgen receptor, ERα or ERβ (IC50, > 10 μM). |
In vivo | AZD7594 has anti-inflammatory activity and efficiently inhibits rat lung edema. AZD5423 displayed a potent inhibition of lung edema in a rat model of allergic airway inflammation following dry powder inhalation. |
Alias | AZD7594, AZ13189620 |
Molecular Weight | 606.62 |
Formula | C32H32F2N4O6 |
Cas No. | 1196509-60-0 |
Smiles | C[C@H](NC(=O)C(C)(F)F)[C@H](Oc1ccc2n(ncc2c1)-c1cccc(c1)C(=O)N[C@@H]1CCOC1)c1ccc2OCCOc2c1 |
Relative Density. | 1.40 g/cm3 (Predicted) |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 79 mg/mL (130.23 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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