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Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $59 | In Stock | |
10 mg | $98 | In Stock | |
25 mg | $189 | In Stock | |
50 mg | $345 | In Stock | |
100 mg | $513 | In Stock |
Description | XCT790 is a potent, selective and inverse agonist of estrogen-related receptor alpha(ERRα). |
Targets&IC50 | ERRα:0.37 μM (IC50) |
Kinase Assay | The inhibition of SHP2 from the tested compounds (SHP099) concentrations varying from 0.003-100 μM is monitored using an assay in which 0.5 nM of SHP2 is incubated with of 0.5 μM of peptide IRS1_pY1172(dPEG8)pY1222. After 30-60 minutes incubation at the surrogate substrate, DiFMUP is added to the reaction and incubated at 25 °C for 30 minutes. The reaction is then quenched by the addition of 5 μL of a 160 μM solution of bpV(Phen). The fluorescence signal is monitored using a microplate reader using excitation and emission wavelengths of 340 nm and 450 nm, respectively[1]. |
Molecular Weight | 596.42 |
Formula | C23H13F9N4O3S |
Cas No. | 725247-18-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO: <1 mg/mL (insoluble or slightly soluble), Sonication and heating are recommended. ![]() |
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