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Cintirorgon

Catalog No. TQ0007 CAS 2055536-64-4

Synonyms: LYC-55716

Purity 98.00% Datasheet

Cintirorgon (LYC-55716) is a selective, oral agonist of RORγ. Cintirorgon modulates gene expression of RORγ expressing T lymphocyte immune cells.

Cintirorgon, CAS 2055536-64-4

Pack Size	Availability	Price/USD
1 mg	Inquiry	86.00
5 mg	Inquiry	167.00
10 mg	Inquiry	230.00
50 mg	Inquiry	716.00
100 mg	Inquiry	1265.00
1 mL * 10 mM (in DMSO)	Inquiry	220.00

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Purity 98.00%

Datasheet MSDS

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Cintirorgon (LYC-55716) is a selective, oral agonist of RORγ. Cintirorgon modulates gene expression of RORγ expressing T lymphocyte immune cells.
Targets&IC50

Synonyms	LYC-55716
Purity	98.00%
Molecular Weight	603.53
Formula	C27H23F6NO6S
CAS No.	2055536-64-4

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

DMSO: 110 mg/mL (182.26 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Lycera Announces Initiation of Phase 1/2a Study ARGON of Immuno-Oncology Candidate LYC-55716 in Patients with Advanced Solid Tumors. Jan 04, 2017.

Related Products

Related compounds with same targets

TAK-828F Xylan Vimirogant AZD-0284 RORγt Inverse agonist 8 A-9758 S18-000003 FM26

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