Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 μM)
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 98.00 | |
5 mg | In stock | $ 247.00 | |
10 mg | In stock | $ 413.00 | |
25 mg | In stock | $ 692.00 | |
50 mg | In stock | $ 985.00 | |
100 mg | In stock | $ 1,330.00 | |
500 mg | In stock | $ 2,660.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 272.00 |
Description | Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 μM) |
Targets&IC50 | σ2 receptor:1239 nM(Ki), σ1 receptor:1.14 nM nM(Ki), ERG (human):1.54 μM |
Molecular Weight | 363.86 |
Formula | C19H23ClFN3O |
CAS No. | 1639220-17-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 12.5 mg/mL (34.35 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Sigma-1 receptor antagonist 3 1639220-17-9 Angiogenesis GPCR/G Protein JAK/STAT signaling Tyrosine Kinase/Adaptors Sigma receptor HER KcsA Potassium Channel inhibit Sigma 1 receptor antagonist 3 Inhibitor σ-1 receptor antagonist 3 Sigma Receptor Sigma1 receptor antagonist 3 inhibitor