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Sigma-1 receptor antagonist 3 is a more potent and selective antagonist of Sigma-1 (σ1) receptor (Ki = 1.14 nM) than σ2 receptor(Ki = 1239 nM). Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG, IC50 = 1.54 μM)
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $81 | In Stock | |
5 mg | $197 | In Stock | |
10 mg | $322 | In Stock | |
25 mg | $529 | In Stock | |
50 mg | $718 | In Stock | |
100 mg | $953 | In Stock |
Description | Sigma-1 receptor antagonist 3 is a potent and selective antagonist of Sigma-1 (σ1) receptor(Ki : 1.14 nM), has the potential for the neuropathic pain. |
Targets&IC50 | σ1 receptor:1.14 nM nM(Ki), ERG (human):1.54 μM , σ2 receptor:1239 nM(Ki) |
Molecular Weight | 363.86 |
Formula | C19H23ClFN3O |
Cas No. | 1639220-17-9 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | DMSO: <1 mg/mL (insoluble or slightly soluble), Sonication is recommended. |
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