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Tetrabenazine Racemate

Catalog No. T3534 CAS 718635-93-9

Synonyms: Nitoman, Ro 1-9569 Racemate, Rubigen, TETRABENAZINE

Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affinity label for the vesicle transport system.

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Tetrabenazine Racemate Chemical Structure

Tetrabenazine Racemate, CAS 718635-93-9

Pack Size	Availability	Price/USD
10 mg	In stock	$ 46.00
25 mg	In stock	$ 83.00
50 mg	In stock	$ 124.00
100 mg	In stock	$ 165.00
200 mg	In stock	$ 216.00

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Purity: 98.86%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high-affinity label for the vesicle transport system.
In vivo	BMS-663068 has good antiviral activity in subjects infected with virus shown to be susceptible (IC50, <100 nM) to the agent[1].

Synonyms	Nitoman, Ro 1-9569 Racemate, Rubigen, TETRABENAZINE
Molecular Weight	317.42
Formula	C19H27NO3
CAS No.	718635-93-9

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 55 mg/mL (173.27 mM)

References and Literature

1. Jankovic, J. and J. Beach, Long-term effects of tetrabenazine in hyperkinetic movement disorders. Neurology, 1997. 48(2): p. 358-62. 2. Kenney, C., C. Hunter, and J. Jankovic, Long-term tolerability of tetrabenazine in the treatment of hyperkinetic movement disorders. Mov Disord, 2007. 22(2): p. 193-7.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library Drug Repurposing Compound Library Anti-Cancer Drug Library Anti-Cancer Approved Drug Library Bioactive Compound Library FDA-Approved Drug Library Human Metabolite Library Anti-Cancer Compound Library Ion Channel Inhibitor Library Bioactive Compounds Library Max

Related Products

Related compounds with same targets

Diclofensine Valbenazine tosylate VMAT2-IN-2 tosylate (+)-Kavain Valbenazine Xanthoangelol Tetrabenazine Reserpine

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Keywords

Tetrabenazine Racemate 718635-93-9 Membrane transporter/Ion channel Monoamine Transporter Nitoman inhibit Inhibitor Ro 1-9569 Ro 1-9569 Racemate Rubigen TETRABENAZINE inhibitor

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